Enzyme modulator
Type of drug
An enzyme modulator is a type of drug which modulates enzymes. They include enzyme inhibitors and enzyme inducers. In an homogeneous assay, "an enzyme modulator ... is covalently linked to the ligand which competes with free ligand from the test sample for the available antibodies."[1]
See also
- Channel modulator
- Receptor modulator
- Transporter modulator
References
- ^ Tijssen, P. (1 August 1985). Practice and Theory of Enzyme Immunoassays. Elsevier. p. 382. ISBN 9780080858845. Retrieved 22 January 2015.
In the homogeneous assay, an enzyme modulator (antibody, inhibitor or receptor for the enzyme) is covalently linked to the ligand which competes with free ligand from the test sample for the available antibodies.
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Receptor/signaling modulators
similar/related
- Amino acids and related: GABA receptor modulators
- GABAA receptor positive modulators
- GABA metabolism and transport modulators
- GHB receptor modulators
- Glutamate metabolism and transport modulators
- Glycine receptor modulators
- Ionotropic glutamate receptor modulators
- Metabotropic glutamate receptor modulators
- Monoamines: Adrenergic receptor modulators
- Dopamine receptor modulators
- Histamine receptor modulators
- Melatonin receptor modulators
- Monoamine metabolism modulators
- Monoamine neurotoxins
- Monoamine releasing agents
- Monoamine reuptake inhibitors
- Serotonin receptor modulators
- hTAAR modulators
- Acetylcholine: Acetylcholine metabolism and transport modulators
- Muscarinic acetylcholine receptor modulators
- Nicotinic acetylcholine receptor modulators
- Others: Imidazoline receptor modulators
- Purine receptor modulators
- Sigma receptor modulators
- Thyroid hormone receptor modulators
- Eicosanoids: Cannabinoid receptor modulators
- Leukotriene signaling modulators
- Prostanoid signaling modulators
- Phospholipids: Lysophospholipid signaling modulators
- PAF receptor modulators
- Steroids: Androgen receptor modulators
- Estrogen receptor modulators
- Glucocorticoid receptor modulators
- Mineralocorticoid receptor modulators
- Progesterone receptor modulators
- Steroid metabolism modulators
- Other nuclear receptors: Aryl hydrocarbon receptor modulators
- Estrogen-related receptor modulators
- FXR and LXR modulators
- PPAR modulators
- Retinoid receptor modulators
- Vitamin D receptor modulators
- Xenobiotic-sensing receptor modulators
- Peptides: Angiotensin receptor modulators
- GH/IGF-1 axis signaling modulators
- GnRH and gonadotropin receptor modulators
- Melanocortin receptor modulators
- Neurokinin receptor modulators
- Opioid receptor modulators
- Oxytocin and vasopressin receptor modulators
- Cytokines: Cytokine receptor modulators
- Chemokine receptor modulators
- Interleukin receptor modulators
- TNF receptor superfamily modulators
- Growth factors: Growth factor receptor modulators
- TGFβ receptor superfamily modulators
non-receptor
- Enzymes: Cytochrome P450 modulators
- Histone deacetylase inhibitors
- Phosphodiesterase inhibitors
- Ion channels: Ion channel modulators
- TRP channel modulators
- Transporters: Sodium-glucose transporter modulators
- Symporter inhibitors
- Others: Nitric oxide signaling modulators
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